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A Convenient Synthesis and Biological Activity of Novel Pyrido[4,3-d]pyrimidin-4(3H)-ones
Ren, Qingyun1; Xia, ShiYan2; Gu, Yucheng1,3; Li, Baoju2; He, Hongwu1
2015
发表期刊JOURNAL OF HETEROCYCLIC CHEMISTRY
ISSN0022-152X
卷号52期号:3页码:647-652
摘要Fifteen novel 2-alkylamino-3-aryl-8-cyano-5-methyl-7-(methylthio)-pyrido[4,3-d]pyrimidin-4(3H)-ones 6a, 6b, 6c, 6d, 6e, 6f, 6g, 6h, 6i, 6j, 6k, 6l, 6m, 6n, 6o were designed and have been successfully synthesized via tandem aza-Wittig and annulation reactions with the corresponding iminophosphoranes 4, aryl isocyanate, and amines in good yields. Their structures were clearly verified by IR spectroscopy, H-1-NMR spectroscopy, EI-MS, and elemental analysis, and in the case of compound 6i, further analyzed by single-crystal X-ray diffraction. The preliminary results of an in vivo bioassay showed that some compounds display moderate antifungal activity.
学科领域Chemistry, Organic
DOI10.1002/jhet.2119
收录类别SCI
语种英语
WOS记录号WOS:000354018900003
出版者WILEY-BLACKWELL
nyguid4024f32e-3446-43c3-9186-370b0489b809
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文献类型期刊论文
条目标识符http://ir.nais.net.cn/handle/2HMLN22E/148849
专题蔬菜花卉研究所_植物保护研究室
通讯作者Ren, Qingyun
作者单位1.Cent China Normal Univ, Coll Chem, Key Lab Pesticide & Chem Biol, Minist Educ, Wuhan 430079, Peoples R China;
2.Chinese Acad Agr Sci, Inst Vegetables & Flowers, Beijing 100081, Peoples R China;
3.Syngenta Jealotts Hill Int Res Ctr, Bracknell RG42 6EY, Berks, England
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Ren, Qingyun,Xia, ShiYan,Gu, Yucheng,et al. A Convenient Synthesis and Biological Activity of Novel Pyrido[4,3-d]pyrimidin-4(3H)-ones[J]. JOURNAL OF HETEROCYCLIC CHEMISTRY,2015,52(3):647-652.
APA Ren, Qingyun,Xia, ShiYan,Gu, Yucheng,Li, Baoju,&He, Hongwu.(2015).A Convenient Synthesis and Biological Activity of Novel Pyrido[4,3-d]pyrimidin-4(3H)-ones.JOURNAL OF HETEROCYCLIC CHEMISTRY,52(3),647-652.
MLA Ren, Qingyun,et al."A Convenient Synthesis and Biological Activity of Novel Pyrido[4,3-d]pyrimidin-4(3H)-ones".JOURNAL OF HETEROCYCLIC CHEMISTRY 52.3(2015):647-652.
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